TABLE 3.
Specific P450 contents (picomoles per milligram microsomal protein) in human small intestinal microsomes (HIM)
| P450 | 1A1 | 2A6 | 2B6 | 2C9 | 2C19 | 2D6 | 2E1 | 2J2 | 3A4 | 3A5 |
|---|---|---|---|---|---|---|---|---|---|---|
| Mean | 5.6 | BLD | BLD | 8.4 | 1.0 | 0.5 | BLD | 0.9 | 43 | 16 |
| (individuals) | ||||||||||
| n | 3 | 31 | 31 | 31 | 31 | 29 | 31 | 31 | 31 | 11 |
| Range | 3.6–7.7 | 2.9–27 | <0.6–3.9 | <0.2–1.4 | <0.2–3.1 | 8.8–150 | 4.9–25 | |||
| Mean ± S.D.a | BLD | BLD | BLD | 11 ± 0.5 | 2.1 ± 0.1 | 0.7 ± 0.01 | BLD | 1.0 ± 0.1 | 58 ± 1.0 | 16 ± 0.3 |
| (pooled HIM)b | ||||||||||
| LOD | 1.5 | 2.0 | 1.3 | 2.0 | 0.6 | 0.2 | 0.2 | 0.2 | 8 | 4 |
BLD, below limit of detection; LOD, limit of detection (picomoles per milligram).
Values denote the mean ± S.D. of triplicate measurements.
The pooled sample consisted of 31 (for P450s 1A1, 2A6, 2B6, 2C9, 2C19, 2D6, 2E1, and 3A4) or 11 (for CYP3A5) individual preparations.