Table 2.
Pharmacology of prostamide antagonists AGN 204396 and AGN 204397
Receptor | 204396 Kb (nM) | AGN 204397 Kb (nM) |
---|---|---|
Prostamide | 2635 | 3099 |
DP1 | NA | NA |
EP1 | NA | NA |
EP2 | NA | NA |
EP3 | NA | NA |
EP4 | NA | NA |
FP | NA | NA |
IP | NA | NA |
TP | 1.5 | 1.5 |
Abbreviation: prostamide, prostaglandin-ethanolamide.
Prostamide refers to activity in the feline iris sphincter preparation; other preparations are human recombinant prostanoid receptors.