Table 1.
Chemical properties of PBR ligands
| Ligands | Ki (nM)* | LogD | cLogD | fP (%) |
|---|---|---|---|---|
| PBR01 | 0.24 | - | 4.4 | - |
| PBR06 | 0.30 | 4.05 | 4.37 | 3.5 |
| PBR28 | 0.59 | 3.01 | 2.95 | 5.6 |
| DAA1106 | 0.21 | - | 4.28 | - |
| PK 11195 | 4.12 | 3.97 | 5.28 | - |
*
Determined with rhesus brain
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