Table II.
168 compounds categorized by BDDCS Class.
| High Solubility | Low Solubility | |||
|---|---|---|---|---|
| Extensive Metabolism | Class 1 | Class 2 | ||
| Abacavir | Ketoprofen | Albendazole | Ketoconazole | |
| Acetaminophen | Ketorolac | Amiodarone | Lansoprazole | |
| Albuterol | Labetolol | Atorvastatin | Lopinavir | |
| Allopurinol | Levamisole | Azathioprine | Lovastatin | |
| Amitryptyline | Levodopa | Azithromycin | Mebendazole | |
| Antipyrine | Lidocaine | Carbamazepine | Mefloquin | |
| Buspirone | Meperidine | Carvedilol | Nalidixic acid | |
| Caffeine | Metoprolol | Chlorpromazine | Naproxen | |
| Chloramphenicol | Metronidazole | Cisapride | Nelfinavir | |
| Chlorpheniramine | Midazolam | Clofazamine | Nevirapine | |
| Codeine | Minocycline | Cyclosporine | Nifedipine | |
| Colchicine | Misoprostol | Danazol | Oxaprozin | |
| Cyclophosphamide | Morphine | Dapsone | Phenytoin | |
| Desipramine | Phenobarbital | Diclofenac | Piroxicam | |
| Dexamethasone | Phenylalanine | Diflunisal | Praziquantel | |
| Diazepam | Prednisolone | Efavirenz | Raloxifene | |
| Diltiazem | Primaquine | Flurbiprofen | Rifampin | |
| Diphenhydramine | Promazine | Glipizide | Ritonavir | |
| Disopyramide | Promethazine | Glyburide | Saquinavir | |
| Doxepin | Propranolol | Griseofulvin | Sirolimus | |
| Enalapril | Pyranzinamide | Haloperidol | Spironolactone | |
| Ergonovine | Quinidine | Ibuprofen | Sulfamethoxazole | |
| Ergotamine | Quinine | Indinavir | Tacrolimus | |
| Ethinyl estradiol | Rosiglitazone | Indomethacin | Tamoxifen | |
| Fluoxetine | Salicyclic acid | Itraconazole | Terfenadine | |
| Glucose | Theophylline | Ivermectin | Warfarin | |
| Hydralazine | Valproic acid | |||
| Imipramine | Verapamil | |||
| Isoniazid | Zidovudine | |||
| Isosorbid dinitrate | ||||
| Poor Metabolism | Class 3 | Class 4 | ||
| Acyclovir | Ganciclovir | Acetazolamide | ||
| Amiloride | Hydrochlorothiazide | Aluminum hydroxide | ||
| Amoxicillin | Lamivudine | Amphotericin | ||
| Atenolol | Levofloxacin | Chlorothiazide | ||
| Atropine | Lisinopril | Chlorthalidone | ||
| Bidisomide | Lithium | Ciprofloxacin | ||
| Bisphosphonates | Lomefloxacin | Colistin | ||
| Captopril | Metformin | Digoxin | ||
| Cefazolin | Methotrexate | Furosemide | ||
| Cetirizine | Metoclopramide | Neomycin | ||
| Chloroquine | Nadolol | Nystatin | ||
| Cimetidine | Neostigmine | Ofloxacin | ||
| Cloxacillin | Penicillins | Phenazopyridine | ||
| Dicloxacillin | Pravastatin | Talinolol | ||
| Doxycycline | Pyridostigmine | |||
| Ephedrine | Ranitidine | |||
| Erythromycin | Riboflavin | |||
| Ethambutol | Tetracycline | |||
| Famotidine | Trimethoprim | |||
| Fexofenadine | Valsartan | |||
| Fluconazole | Zalcitabine | |||
| Folinic acid | ||||