Table II.
168 compounds categorized by BDDCS Class.
High Solubility | Low Solubility | |||
---|---|---|---|---|
Extensive Metabolism | Class 1 | Class 2 | ||
Abacavir | Ketoprofen | Albendazole | Ketoconazole | |
Acetaminophen | Ketorolac | Amiodarone | Lansoprazole | |
Albuterol | Labetolol | Atorvastatin | Lopinavir | |
Allopurinol | Levamisole | Azathioprine | Lovastatin | |
Amitryptyline | Levodopa | Azithromycin | Mebendazole | |
Antipyrine | Lidocaine | Carbamazepine | Mefloquin | |
Buspirone | Meperidine | Carvedilol | Nalidixic acid | |
Caffeine | Metoprolol | Chlorpromazine | Naproxen | |
Chloramphenicol | Metronidazole | Cisapride | Nelfinavir | |
Chlorpheniramine | Midazolam | Clofazamine | Nevirapine | |
Codeine | Minocycline | Cyclosporine | Nifedipine | |
Colchicine | Misoprostol | Danazol | Oxaprozin | |
Cyclophosphamide | Morphine | Dapsone | Phenytoin | |
Desipramine | Phenobarbital | Diclofenac | Piroxicam | |
Dexamethasone | Phenylalanine | Diflunisal | Praziquantel | |
Diazepam | Prednisolone | Efavirenz | Raloxifene | |
Diltiazem | Primaquine | Flurbiprofen | Rifampin | |
Diphenhydramine | Promazine | Glipizide | Ritonavir | |
Disopyramide | Promethazine | Glyburide | Saquinavir | |
Doxepin | Propranolol | Griseofulvin | Sirolimus | |
Enalapril | Pyranzinamide | Haloperidol | Spironolactone | |
Ergonovine | Quinidine | Ibuprofen | Sulfamethoxazole | |
Ergotamine | Quinine | Indinavir | Tacrolimus | |
Ethinyl estradiol | Rosiglitazone | Indomethacin | Tamoxifen | |
Fluoxetine | Salicyclic acid | Itraconazole | Terfenadine | |
Glucose | Theophylline | Ivermectin | Warfarin | |
Hydralazine | Valproic acid | |||
Imipramine | Verapamil | |||
Isoniazid | Zidovudine | |||
Isosorbid dinitrate | ||||
Poor Metabolism | Class 3 | Class 4 | ||
Acyclovir | Ganciclovir | Acetazolamide | ||
Amiloride | Hydrochlorothiazide | Aluminum hydroxide | ||
Amoxicillin | Lamivudine | Amphotericin | ||
Atenolol | Levofloxacin | Chlorothiazide | ||
Atropine | Lisinopril | Chlorthalidone | ||
Bidisomide | Lithium | Ciprofloxacin | ||
Bisphosphonates | Lomefloxacin | Colistin | ||
Captopril | Metformin | Digoxin | ||
Cefazolin | Methotrexate | Furosemide | ||
Cetirizine | Metoclopramide | Neomycin | ||
Chloroquine | Nadolol | Nystatin | ||
Cimetidine | Neostigmine | Ofloxacin | ||
Cloxacillin | Penicillins | Phenazopyridine | ||
Dicloxacillin | Pravastatin | Talinolol | ||
Doxycycline | Pyridostigmine | |||
Ephedrine | Ranitidine | |||
Erythromycin | Riboflavin | |||
Ethambutol | Tetracycline | |||
Famotidine | Trimethoprim | |||
Fexofenadine | Valsartan | |||
Fluconazole | Zalcitabine | |||
Folinic acid |