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. 2003 Oct;12(10):2173–2182. doi: 10.1110/ps.03171903

Table 1.

Values of Kd from previous studies

Reference Protease pH Kd τ1/2 (sec) Remark
Holzman et al. 1991 HIV-2 4.5 87 μM
7.5 28 μM
Grant et al. 1992 HIV-1 5.0 <10 nM
Towler et al. 1998 HIV-1 7.0 9 μM
HERV-K10 7.0 52.5 μM
Xie et al. 1999 HIV-1 7.0 52.7 μM Autolysis products interferred, Kd taken as upper limit
Stříšovský et al. 2000 HIV-1 6.0 77 μM
Cheng et al. 1990 HIV-1 7.0 50 nM 198
Zhang et al. 1991 HIV-1 3.6 nM Very fast processes assumed
Jordan et al. 1992 HIV-1 <1 nM
HIV-2 <1 nM
Darke et al. 1994 HIV-1 6.5 16 nM Fluorogenic inhibitor used
7.0 39 nM
Pargellis et al. 1994 HIV-1 5.5 5.2 nM 533 0 M NaCl
4.0 nM 745 1.5 M NaCl
Kuzmič et al. 1993 HIV-1 6.4 440 nM 23.9
Uhlíková et al. 1996 HIV-1 6.4 112 nM Integral kinetics
4.5 19 nM

The top part of the table shows the results of sedimentation studies; the bottom part the results of kinetic assays. τ1/2 is the halftime of dimer dissociation.