Table 1.
Water Solubility | T 1/2 (h) | IC50 (ng/mL) | |||
---|---|---|---|---|---|
Compound | mg/ml | pH 7 | Plasma | MCF-7 | EVSA-T |
PTX | 0.01 | <3 | <3 | ||
6 | 0.2 | >24 | 20 | <3 | <3 |
7 | 0.6 | No PTX | 4 | <3 | <3 |
8 | 0.5 | No PTX | No PTX | 69 | 59 |
Water Solubility | T 1/2 (h) | IC50 (ng/mL) | |||
---|---|---|---|---|---|
Compound | mg/ml | pH 7 | Plasma | MCF-7 | EVSA-T |
PTX | 0.01 | <3 | <3 | ||
6 | 0.2 | >24 | 20 | <3 | <3 |
7 | 0.6 | No PTX | 4 | <3 | <3 |
8 | 0.5 | No PTX | No PTX | 69 | 59 |