Table 2. Summary of changes in angiogenic factors compared with patient outcome.
| Agent | Pata | Outcome | Fluidb | VEGF | bFGF | VCAM-1 | v-WF | Thmc | Esel | uPAsr | MMP-2 | MMP8 | MMP9 | TIMP1 | TIMP2 |
| Razoxane | 35 | StD(11) | U, P, S (56) | S, Pre PD>StDd | S, Post PD>StDd | S, Post PD>StDd | S, Pre PD>StDd | P, Pre PD>StDd | |||||||
| U, PD Pre vs Poste | U, Pre PD>StDd | S, PD Pre vs Poste | S, Post PD>StDd | P, Post PD>StDd | |||||||||||
| MM1270 | 75 | StD(19) | P(28) | Nc | w/AUCe | Nc | w/AUCe | Nc | W/Cmaxe | W/AUCe | W/AUCe | ||||
| BAY 12-9566 | 21 | No response | P(29) | Nc | Nc | Post>Pre | |||||||||
| COL-3 | 35 | StD(8) | S, P(28) | S, Nc | S, Nc | P, Post PD>StD | P, Nc | ||||||||
| Endostatin | 25 | StD(1), MR(1) | S(28,56) | Nc | Nc | Nc | Nc | ||||||||
| TNP-470 | 12 | No response | U, S(28) | Nc | S, Nc | Nc | |||||||||
| SU5416 | 22 | StD(3), MR(1) | U(36) | Pre>Poste | Nc | ||||||||||
| Thalidomide | 16 | PR(2), MR(2), StD(12) | S, U(56) | Nc | S, Decreased, U, Nc |
Patients studied.
P=Plasma, S=Serum, U=Urine (days post-treatment).
Thrombomodulin.
Significant differences.
Significant increase. Nc=no significant change; Pre=before treatment; Post=after treatment; PD=progressive disease; StD=stable disease; MR=minor response; PR=partial response; AUC=area under concentration curve.