. Author manuscript; available in PMC: 2008 Jun 26.

Published in final edited form as: Biochemistry. 2007 Nov 29;46(51):15089–15102. doi: 10.1021/bi7018783

Table 4.

ADP Reversal of Inhibition of the Various Compounds^a

compound	[drug] (µM)	activation (%)	K_act ADP (µM)	R²
no drug		21 (1.3)	17 (6.2)	0.88
GW5074	4	21 (9.4)	449 (411)	0.71
GW5074	8	34 (2.0)	31 (9.2)	0.90
hexachlorophene	3	92 (4.4)	89 (15)	0.97
ATA	8	207 (17)	222 (49)	0.96
bithionol	10	164 (4.7)	51 (6.2)	0.98
BSB	15	79 (1.8)	41 (32)	0.99
BH3I	10	140 (5.9)	34 (7.0)	0.95
DES	8	64 (2.0)	19 (3.4)	0.96

Shown here is a summary of the data shown in Figure 9, fitted to eq 6.