TABLE 2.
Pharmacokinetic results for BPR after a single s.c. dose in immunocompromised, infected BALB/c micea
| Dosing regimen (mg/kg) | Cmax (mg/liter) | Tmax (h) | AUC0-∝ (mg·h/liter) | VF (liter/kg) | Half-life (h) | CL (ml/h/kg) |
|---|---|---|---|---|---|---|
| 1 | 1.74 | 0.48 | 1.84 | 0.19 | 0.25 | 0.54 |
| 2.5 | 2.91 | 0.41 | 2.57 | 0.63 | 0.45 | 0.97 |
| 10 | 19.75 | 0.15 | 15.79 | 0.38 | 0.42 | 0.63 |
| 25 | 38.59 | 0.47 | 35.25 | 0.41 | 0.40 | 0.71 |
Tmax, time required to achieve Cmax; AUC0-∝, AUC from time zero to infinity; VF, volume of distribution; CL, clearance.