Table 1.
Spectrally Determined Binding Constants for Flurbiprofen, in the Absence and Presence of Dapsone, Obtained with CYP2C9.1, CYP2C9.2, CYP2C9.3 and CYP2C9.5 Enzymes.
| Enzyme | No Dapsone KS (μM) | + Dapsone KS (μM) |
|---|---|---|
| CYP2C9.1 | 7.5 | 2.8 |
| CYP2C9.2 | 4.5 | 1 |
| CYP2C9.3 | 13.8 | 3 |
| CYP2C9.5 | 16 | 3 |