TABLE 3.
Summary of single channel conductances (g) and mean channel lifetimes (τ) for 1-Me-Trp gA analogues
Conditions were as follows: diphytanoylphosphatidylcholine, 1 m salt, 200 mV, 25 °C.
Analogue | ga | τ | Salt |
---|---|---|---|
picosiemens | ms | ||
gA | 47 | 680 | CsCl |
[1-Me-Trp9]gA | 45 | 770 | CsCl |
[1-Me-Trp11]gA | 43 | 1200 | CsCl |
[1-Me-Trp13]gA | 50 | 790 | CsCl |
[1-Me-Trp15]gA | 51 | 870 | CsCl |
[1-Me-Trp9,11]gA | 39 | 1300 | CsCl |
[1-Me-Trp13,15]gA | 47 | 940 | CsCl |
[1-Me-Trp9,11,13,15]gA | 36 | 2200 | CsCl |
gA | 15.0b | 840b | NaCl |
[1-Me-Trp9]gA | 12.0 | 730 | NaCl |
[1-Me-Trp15]gA | 14.5 | 830 | NaCl |
[Phe9]gA | 6.0b | 1000b | NaCl |
[Phe15]gA | 10.9b | 790b | Nacl |
S.E. of measurement: ± 0.5 - 1.0 picosiemens.
Data from Ref. 27 are shown for comparison.