Table 2.
Investigation of Heterocycle Scope
Entry | Heterocycle | Time (h) | # | Yield (%)a |
---|---|---|---|---|
1 | ![]() |
14 | 3 | 59 |
2 | 14 | 4 | 83 | |
3 | 24 | 5 | 64 | |
4 | ![]() |
14 | 6 | 96 |
5 | 9.5 | 7 | 98 | |
6 | 7 | 8 | 96 |
Isolated yield of pure product.
Investigation of Heterocycle Scope
Entry | Heterocycle | Time (h) | # | Yield (%)a |
---|---|---|---|---|
1 | ![]() |
14 | 3 | 59 |
2 | 14 | 4 | 83 | |
3 | 24 | 5 | 64 | |
4 | ![]() |
14 | 6 | 96 |
5 | 9.5 | 7 | 98 | |
6 | 7 | 8 | 96 |
Isolated yield of pure product.