Table 43.
entry | ligand | conv. (%) | b/l | ee (%) | config. |
---|---|---|---|---|---|
1 | (2R,4R)-Chiraphite | 32 | 10.8 | 51 | R |
2 | (R,S)-BINAPHOS | 35 | 4.6 | 81 | R |
3 | (S,S)-Kelliphite | 32 | 9.2 | 3 | S |
4 | diazaphospholane | 73 | 5.7 | 80 | R |
5 | (R,R)-Ph-BPE | 33 | 45 | 92 | R |
6 | (2R,4R)-Chiraphite | 74 | 5.8 | 13 | R |
7 | (R,S)-BINAPHOS | 58 | 2.1 | 68 | R |
8 | (S,S)-Kelliphite | 99 | 10.1 | 66 | S |
9 | diazaphospholane | 100 | 3.9 | 80 | R |
10 | (R,R)-Ph-BPE | 67 | 7.6 | 90 | R |
11 | (2R,4R)-Chiraphite | 34 | 204 | 50 | R |
12 | (R,S)-BINAPHOS | 23 | 7.1 | 58 | S |
13 | (S,S)-Kelliphite | 32 | 100 | 75 | R |
14 | diazaphospholane | 92 | 47 | 95 | S |
15 | (R,R)-Ph-BPE | 34 | 263 | 82 | S |