Table 5.
Enzyme | Km(ATP) (μM) | Fold Inflation | Kd(ATP) (μM) c | Fold Inflation |
---|---|---|---|---|
WT | 107±14 | - | 30±3 | - |
R141M | 5200±474b | 49 | 816±160 | 27 |
Spectrophotometric assays were performed in 100 mM MOPS, 200 mM KCl, 1 mM DTT (pH 7.0) in the presence of 10 mM MgCl2 at 30°C. [ATP] was kept saturating (5 mM). Errors represent the standard error of the fit.
Assays contained 20 mM MgCl2.
Determined by tryptophan fluorescence. Averaged data points from 3 [protein] were fit to a two site model using the equation y = Bmax1[X]/(Kd1 + [X]) + Bmax2[X]/(Kd2 + [X]).
Kd2 values (WT: 14 mM, R141M: 41 mM) are too weak to be physiologically relevant and are not considered in the comparison. Errors represent the standard error of the fit.