Table 5.
Hydrosilylation of alkynyl carbonyl compounds.
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---|---|---|---|---|---|---|---|
entry | alkyne | cmpd | silane | mol% 7 | product | yield | selectivityb |
1 |
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77 | BnMe2SiH | 0.5 | 78 | 98 | >20:1 |
2 | 77 |
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5 | 80 | 89 | >20:1 | |
3 |
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81 | (allyl)Me2SiH | 4 | 82 | 81 | >20:1 |
4 |
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84 | PhMe2SiH | 2 | 85 | 96 | >20:1 |
5 | 84 | (EtO)3SiH | 1 | 86 | 99 | 5:1 | |
6 |
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87 | BnMe2SiH | 1 | 88 | 67 (89)c | >20:1 |
7 |
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89 | BnMe2SiH | 1 | 90 | 88 | 7:1 |
8 |
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91 | (allyl)Me2SiH | 5 | 92 | 72 | 15:1 |
9 |
![]() |
93 | BnMe2SiH | 3 | 94 | 34 | >20:1 |
10 |
![]() |
95 | BnMe2SiH | 1 | 96 | 94 | >20:1 |
Reactions performed using 1.2 eq. silane at 0.5 M in acetone for 30 min.
Ratio of β-vinylsilane: α-vinylsilane determined by analysis of crude 1H NMR. In all cases only (Z)-vinylsilane isomers were observed.
Yield in parenthesis is based on recovered alkyne.