Table 3.
Purification Schemes for Five Recombinant Human Dihydrodiol Dehydrogenase (AKR) Isoforms a
protein | purification step | volume (mL) | total protein (mg) | total activity (:mol min-1 mg-1) | specific activity (:mol min-1 mg-1) | purification factor (-fold) | yield (5%) |
---|---|---|---|---|---|---|---|
AKR1A1 | sonicate | 70 | 470 | 668 | 1.42 | 1 | 100 |
DE52 cellulose | 12.5 | 88.5 | 233 | 2.63 | 1.85 | 34.7 | |
Blue-Sepharose | 7.1 | 30.5 | 183 | 6.0 | 4.23 | 27.4 | |
AKR1C1 | sonicate | 61 | 460 | 59 | 0.13 | ||
DE52 cellulose | 16 | 23 | 46 | 2.0 | 15 | 78 | |
Blue Sepharose | 8 | 20 | 42 | 2.1 | 16 | 71 | |
AKR1C2 | sonicate | 77 | 510 | 42 | 0.08 | ||
DE52 cellulose | 18 | 19 | 39 | 2.1 | 25 | 93 | |
Blue-Sepharose | 11 | 15 | 37 | 2.5 | 31 | 88 | |
AKR1C3 | sonicate | 51 | 310 | 65 | 0.21 | ||
DE52 cellulose | 56 | 25 | 51 | 2.0 | 10 | 78 | |
Blue-Sepharose | 5 | 12 | 34 | 2.8 | 13 | 52 | |
AKR1C4 | sonicate | 44 | 270 | 4.6 | 0.02 | ||
DE52 cellulose | 12 | 23 | 2.8 | 0.12 | 6 | 61 | |
Blue-Sepharose | 8 | 13 | 2.7 | 0.21 | 11 | 59 |
Specific activities throughout the purifications were measured using 75 :M androsterone (AKR1C4) or 1 mM 1-acenaphthenol (AKR1C1-AKR1C3) as the substrate in reaction mixtures containing 100 mM KPO4 (pH 7.0) and 2.3 mM NAD+ at 25.0 °C.