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. 2008 Oct 15;105(43):16809–16813. doi: 10.1073/pnas.0805677105

Table 1.

In vitro activity data for BI-78D3 and related compounds

Molecule ID MW DELFIA assay data LanthaScreenTM kinase assay data
graphic file with name zpq99908529000g1.jpg BI-78D3* 379.37 IC50 = 500 nM IC50 = 280 nM
graphic file with name zpq99908529000g2.jpg BI-83C9 321.33 IC50 = 237 nM IC50 = 3.1 μM
graphic file with name zpq99908529000g3.jpg BI-83C7 306.32 IC50 = 183 nM IC50 = 3.3 μM
graphic file with name zpq99908529000g4.jpg BI-83C8 319.36 IC50 = 7.5 μM No Inhibition at 100 μM
graphic file with name zpq99908529000g5.jpg BI-83B3 268.33 No Displacement at 25 μM No Inhibition at 100 μM
graphic file with name zpq99908529000g6.jpg BI-83C11 378.38 No Displacement at 25 μM No Inhibition at 100 μM