Table 3.
Compound | IC50 (μM) | Solubility in saline (μM) | % Cell viability | |
---|---|---|---|---|
20 μM | 50 μM | |||
CFTRinh-172 | 0.38 ± 0.04 | 17 | 86 | not soluble |
Tetrazolo-172 | 0.76 ± 0.2 | 189 | 87 | 73 |
Oxo-172 | 1.4 ± 0.2 | 420 | 93 | 91 |
α-Me-172 | 8.2 ± 0.4 | 259 | 89 | 72 |
Pyridine-NO-172 | 8.7 ± 0.7 | 264 | not determined |