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. Author manuscript; available in PMC: 2008 Dec 4.
Published in final edited form as: Org Lett. 2007 Jan 18;9(2):203–206. doi: 10.1021/ol062610v

Table 3.

Cross-Coupling of Potassium β-Aminoethyltrifluoroborate 1a with Electron-Poor Aryl Bromides

graphic file with name nihms60272f4.jpg
entry Ar-X % isolated yield
1 graphic file with name nihms60272t7.jpg 2a, 90
2 graphic file with name nihms60272t8.jpg 2b, X = Br, 82
X = I, 79
X = Otf, 77
3 graphic file with name nihms60272t9.jpg 2c, 79
4 graphic file with name nihms60272t10.jpg 2d, 84
5 graphic file with name nihms60272t11.jpg 2e, 84
6 graphic file with name nihms60272t12.jpg 2f, 73
7 graphic file with name nihms60272t13.jpg 2g, 74
8 graphic file with name nihms60272t14.jpg 2h, 79
9 graphic file with name nihms60272t15.jpg 2i, 85
10 graphic file with name nihms60272t16.jpg 2j, 79