Table 3.
Reaction constants of the designed peptides for p38α
Peptide | KM or KMapp (μM) | kcat or kcatapp (min−1) | kcatapp/KMapp (μM−1 min−1) |
---|---|---|---|
ERKSub | 1200 + 600 | 570 + 185 | 0.5 |
MEK1ERK | 65 + 14 | 570 + 28 | 8.7 |
MEK2ERK | 30 + 10 | 1000 + 42 | 33 |
Reaction constants of the designed peptides for p38α
Peptide | KM or KMapp (μM) | kcat or kcatapp (min−1) | kcatapp/KMapp (μM−1 min−1) |
---|---|---|---|
ERKSub | 1200 + 600 | 570 + 185 | 0.5 |
MEK1ERK | 65 + 14 | 570 + 28 | 8.7 |
MEK2ERK | 30 + 10 | 1000 + 42 | 33 |