Table 1.
EC50 values for various PAQR ligands.
log EC50 pM (EC50) | ||
---|---|---|
Adiponectin | Progesterone | |
AdipoR1 | −0.13 ± 0.08 (0.7 pM) |
N.R. |
AdipoR2 | −0.38 ± 0.17 (2.4 pM) |
N.R. |
mPRγ | N.R. | 3.11 ±0.44 (1.3 nM) |
PAQR6 | N.R. | 3.42 ± 0.88 (2.6 nM) |
mPRα | N.R. | 3.36 ± 0.08 (2.3 nM) |
mPRβ | N.R. | 3.21 ± 0.61 (1.6 nM) |
PAQR9 | N.R. | 4.14 ± 0.86 (13.8 nM) |
N.R. No response