Table 1.
TGF-β isoform | GC-1008 (n = 6) |
---|---|
TGF-β1 (40 pM) | 1 ± 2 |
TGF-β2 (40 pM) | 14 ± 5 |
TGF-β3 (40 pM) | 7 ± 2 |
IC50 values are given in nM. KD values for GC-1008 against TGF-β 1 and 3 have been determined in a competition assay with TGF-β receptor type II to be 50 pM and 250 pM, respectively.