Table 2.
Protein | KD, (nM)1 TMEGF45 | KM,TM(nM) TMEGF45 | KM,PC(∝M) TMEGF45 | kcat(s-1) TMEGF45 |
---|---|---|---|---|
wild type | 68 | 140±12 | 0.32±0.1 | 5.0±0.1 |
D349N | 43 | 440±38 | 0.77±0.2 | 0.69±0.01 |
E357Q | 55 | 149±29 | 1.0±0.2 | 0.36±0.06 |
E357D | ND | 542±41 | 0.62±0.26 | 0.22±0.02 |
Y358A | ND | 623±100 | 1.3±0.3 | 0.08±0.003 |
Y358H | ND | 163±16 | 1.6±0.16 | 0.2±0.02 |
Y358W | ND | 61±9 | 0.8±0.5 | 5.6±1.6 |
F376W | ND | 208±19 | 0.9±0.14 | 15±4 |
M388L | 57 | 140±40 | 0.38±0.1 | 7.8±0.5 |
D400N | ND | 616±131 | 0.7±0.04 | 0.04±0.001 |
D400E | 49 | 237±16 | 1.36±0.1 | 0.17±0.01 |
Kd was determined by Scatchard analysis of the fluorescein-EGR-chloromethylketone-labeled thrombin binding data.