Table 3.
Cytotoxicity of compounds 87–89.
| Cell line | 87 IC50 [μM] | 88 IC50 [μM] | 89 IC50 [μM] |
|---|---|---|---|
| HL-60 | 0.01 | 5.73 | 0.08 |
| HL-60/RV+ | 0.19 | 40.30 | 0.80 |
| JURKAT | 0.03 | 12.01 | 0.19 |
| ALL3 | <0.01 | 4.24 | 0.16 |
| NCEB1 | 0.06 | 39.24 | 0.50 |
| JEKO | 0.08 | 25.1 | 0.56 |
| MOLT3 | 0.01 | 6.41 | 0.06 |
| SKNLP | <0.01 | 10.04 | 0.11 |
| Y79 | >100 | >100 | >100 |
| PC9 | 0.04 | 11.29 | 0.13 |
| TC71 | 0.03 | 24 | 0.20 |
| HTB-15 | 0.10 | 58 | 0.50 |
| WD0082 | 0.05 | 11 | 0.20 |