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. Author manuscript; available in PMC: 2009 Jan 28.
Published in final edited form as: Chemistry. 2008;14(14):4293–4306. doi: 10.1002/chem.200701998

Table 3.

Cytotoxicity of compounds 8789.

Cell line 87 IC50 [μM] 88 IC50 [μM] 89 IC50 [μM]
HL-60 0.01 5.73 0.08
HL-60/RV+ 0.19 40.30 0.80
JURKAT 0.03 12.01 0.19
ALL3 <0.01 4.24 0.16
NCEB1 0.06 39.24 0.50
JEKO 0.08 25.1 0.56
MOLT3 0.01 6.41 0.06
SKNLP <0.01 10.04 0.11
Y79 >100 >100 >100
PC9 0.04 11.29 0.13
TC71 0.03 24 0.20
HTB-15 0.10 58 0.50
WD0082 0.05 11 0.20