Table 3.
Cytotoxicity of compounds 87–89.
Cell line | 87 IC50 [μM] | 88 IC50 [μM] | 89 IC50 [μM] |
---|---|---|---|
HL-60 | 0.01 | 5.73 | 0.08 |
HL-60/RV+ | 0.19 | 40.30 | 0.80 |
JURKAT | 0.03 | 12.01 | 0.19 |
ALL3 | <0.01 | 4.24 | 0.16 |
NCEB1 | 0.06 | 39.24 | 0.50 |
JEKO | 0.08 | 25.1 | 0.56 |
MOLT3 | 0.01 | 6.41 | 0.06 |
SKNLP | <0.01 | 10.04 | 0.11 |
Y79 | >100 | >100 | >100 |
PC9 | 0.04 | 11.29 | 0.13 |
TC71 | 0.03 | 24 | 0.20 |
HTB-15 | 0.10 | 58 | 0.50 |
WD0082 | 0.05 | 11 | 0.20 |