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. 2008 Jul 16;9(7):1276–1320. doi: 10.3390/ijms9071276

Table 5.

Examples for delivery of siRNAs.

Cargo CPP/delivery system proposed uptake mechanism Reference
siRNA MPG, MPGΔNLS (non-covalent) non-endocytotic [131]
siRNA penetratin, transportan n. d. [104]
siRNA Tat47–57, Tat-derived oligocarbamate n. d. [90]
siRNA penetratin n. d. [230]
siRNA H3K8b, H3K8b(+RGD) endocytotic [172]
siRNA stearyl-R8 endocytotic [232]
siRNA Chol-R9 endocytotic [121]
siRNA MPGα endocytotic [236]
siRNA R8-MEND (siRNA/stearyl-R8core) endocytotic [187]
siRNA EB1, MPGΔNLS, bPrPp endocytotic [76]
siRNA Tat48–60, penetratin endocytotic [106]
siRNA RVG peptide n. d. [234]
siRNA rCPP endocytotic [181]