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. 2008 Mar;6(1):21–38. doi: 10.2174/157015908783769680

Table 4.

Antagonists for TRPV1, TRPV2, TRPA1, TRPM8, TRPV3 and TRPV4

ThermoTRP Antagonists
TRPV1 capsazepine; ruthenium red; diphenyltetrahydrofuran (DPTHF); iodo-RTX; SB705498; SB366791; BCTC; NGD-8243; AMG-517; AMG-9810; A-425619; KJM429; JYL1421; JNJ17203212; NGX-4010; WL-1001; WL-1002; A-4975; GRC-6127; 2-(4-pyridin-2-ylpiperazin-1-yl)-1H-benzo[d]imidazole compound 46ad; 6-aryl-7-isopropylquinazolinones; 5,6-fused heteroaromatic urea A-425619.0; 4-aminoquinazoline; halogenated thiourea compounds 23c and 31b; N-tetrahydroquinolinyl, N-quinolinyl and N-isoquinolinyl carboxamides; pentacyclic triterpene; oleanolic acid;
TRPV2 ruthenium red; diphenyltetrahydrofuran (DPTHF)
TRPA1 ruthenium red; camphor; menthol; compoud A and compound B (Abbott Laboratories)
TRPM8 capsazepine; BCTC; CTPC; SB-452533; 2-APB; URB597; cinnamaldehyde
TRPV3 ruthenium red; diphenyltetrahydrofuran (DPTHF)
TRPV4 ruthenium red