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. 2009 Feb 14;65(Pt 3):236–241. doi: 10.1107/S1744309109002267

Table 2. K i values for various ligands to inhibit the binding of [3H]-LY341495 to the N414/439Q mutant of mGluR3 ECD.

Ligand Ki (µM) 95% confidence interval (µM)
LY341495 0.120 0.0909–0.159
DCGIV 0.784 0.658–0.934
L-Glutamate 1.36 1.12–1.65
2R,4R-APDC 24.1 18.9–30.8
1S,3S-ACPD 110 95.7–126
1S,3R-ACPD 146 114–187