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. Author manuscript; available in PMC: 2009 Nov 27.
Published in final edited form as: J Med Chem. 2008 Nov 27;51(22):7205–7215. doi: 10.1021/jm800825n

Table 2.

STD NMR screening of compounds (500 μM) from MORDOR-ranked list of compounds for binding to hTR-P2b (25 μM).

STD NMR Count Percent
Insoluble, causes precipitation or aggregation, insufficiently pure 58
No binding 7 13%
Weak binding 17 31%
Medium binding 14 25%
Strong binding 17 31%
TOTAL 113 100%