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. Author manuscript; available in PMC: 2010 Mar 1.
Published in final edited form as: Expert Opin Pharmacother. 2009 Mar;10(4):555–577. doi: 10.1517/14656560902731993

Table 3.

Reports from Japan of Neisseria gonorrhoeae isolates with elevated MICs to third-generation cephalosporins.

Author, publication year Location Year of Specimen Collection Criteria and Number of isolates assessed Cephalosporin MICs mg/L (range) Comment
Japan
Yamaguchi 1998105 Several Areas of Japan 1991 and 1996 All isolates:
27
Cefpodoxime MIC90=4
Cefditoren MIC90=4
In vitro study of investigational antimicrobial.
Akasaka 2001104 Kitakyushu 1999 Cefdinir Treatment Failure:
2
Cefpodoxime MIC = 4
Cefdinir MIC = 1
Ceftriaxone MIC=0.125
Case report.
Muratani 2001106 Kitakyushu 1999 Cefozopran ≥ 8:
17 of 54
For 17 isolates:
Ceftriaxone MIC90=0.125 (0.03–0.25)
Cefpodoxime MIC90=4 (0.5–4)
Cefixime MIC90=0.5 (0.125–0.5)
Ito 2004107 Central Japan 1999–2000
2001
2002
Cefixime ≥0.5:
0 of 91
39 of 150
67 of 221
1999:
Cefixime MIC90 = 0.06 (≤0.004–0.125)
Ceftriaxone MIC90 = 0.03 (≤0.004–0.06)
2002:
Cefixime MIC90 = 0.5 (≤0.004–2)
Ceftriaxone MIC90 = 0.06 (≤0.004–0.5)
Emerging cefixime resistance.
Ameyama 2002108 Tokyo 2000
2001
Cefixime ≥ 0.25:
9 of 53
4 of 24
2000 and 2001:
Cefixime MIC90 = 0.25
Ceftriaxone MIC90 = 0.06
Report also described a mosaic penA gene among isolates with cefixime MIC ≥0.25.
Tanaka 2002103 Fukuoka City 1995
2000
Cefixime ≥ 0.5
0 of 55
5 of 100
1995:
Cefixime MIC90 = 0.015 (0.002–0.06)
Ceftriaxone MIC90 = 0.015 (0.001–0.03)
2000:
Cefixime MIC90 = 0.25 (0.002–0.5)
Ceftriaxone MIC90 = 0.06 (0.002–0.5)
Emerging cefixime resistance.
Tanaka 2006109 Fukuoka City 2000–2001 Ceftriaxone = 0.5:
1 of 398
Cefixime MIC = 0.5 Analysis of 1 ceftriaxone resistant isolate with mosaic penA and mtrR, ponA, penB mutations.
Yokoi 2007110 Toyota 2002–2003 Cefixime Treatment Failure:
4
Cefixime (0.5–1)
Ceftriaxone (0.125–0.5)
Case report.
Osaka 2006111 Tokyo 2006 Cefixime ≥0.125:
17 of 47
Cefixime MIC90 = 0.125 (0.004–0.25)
Ceftriaxone MIC90 = 0.06 (0.002–0.125)
MIC values compared to those of Ameyama in 2001.
Takahata 2006112 Tokyo 2006 Cefixime ≥ 0.125
28 of 58
For 28 isolates with mosaic penA gene:
Cefixime MIC90 = 0.5 (0.12–0.5)
Ceftriaxone MIC90 = 0.12 (0.016–0.12)
Cefixime MICs correlated with presence of mosaic penA.
Europe
Olsen 2008125 Sweden 2002–2005 Cefixime MIC >0.06–≤0.5:
6 of 679
All had ceftriaxone MIC < 0.125
Hoffmann 2005126 Denmark 2004 Ceftriaxone MIC >0.023 <0.094
81 of 434
No PenA sequencing performed. Serotype, NG-MAST sequence type were related within group of ceftriaxone MIC >0.023 and <0.094
Martin 200651 Europe (ESSTI) 2004 Ceftriaxone > 0.125:
3 of 965
Ceftriaxone MIC = 0.25 Surveillance report. Resistant isolates included 2 from Italy and 1 from Sweden.
Vazquez 2007127 Spain 2004–2005 204 isolates Ceftriaxone MIC90=0.007 (≤0.007–0.12)
Cefditoren MIC90=0.12 (≤0.007–0.25)
Tzelepi 2008128 Greece Dec 2006–Jan 2008 Cefotaxime MIC 0.25–1:
17 of 195
Ceftriaxone MIC90= 0.125 (0.064–0.125)
Cefixime MIC90=0.25 (0.125–0.25)
Isolates were part of a cluster with related serotypes and PFGE patterns in Northern Greece. Isolates were multidrug resistant including penicillin, tetracycline, and fluoroquinolones.
Gonococcal Resistance to Antimicrobials Surveillance Programme 200828 United Kingdom 2007 Cefixime MIC = 0.25:
2 of 1113
Ceftriaxone MIC = 0.015 Surveillance Report.
Australia
Tapsall 2008113 Australia 1997–2006 Ceftriaxone MIC 0.06–0.5:
134 of ~15,000
Isolates with elevated ceftriaxone MIC mostly from travelers or contacts.
Australian Gonococcal Surveillance Program 2008114 Australia 2007 Ceftriaxone MIC 0.06–0.25:
25 of 3,042
Surveillance report.
Elsewhere in Asia
Ray 2005123 Chennai, India
Hyderabad, India
Nagpur, India
Pune, India
Kolkata, India
Bangladesh
2001
2001
2001
2001
2001
1999–2000
Ceftriaxone LS (disk diffusion):
4 of 80
9 of 46
10 of 74
4 of 37
4 of 58
2 of 110
Resistant isolates not confirmed at regional reference laboratory.
Bala 2007124 New Delhi, India 2002–2006 Ceftriaxone MIC≥0.06:
9 of 382
Ceftriaxone MIC 0.064–0.094 No treatment failures reported.
Ye 2002116 China (various) 1993–1998 Ceftriaxone R (not defined):
16 of 2801
Results not confirmed at national reference laboratory.
Guoming 2000117 Zhanjiang, China 1998–1999 Ceftriaxone MIC ≥1:
15 of 98
Ceftriaxone MIC ≥0.06:
34 of 98
Ceftriaxone MIC90=2 (0.016–2)
Wong 2008118 Taipei, Taiwan Apr 2006–Aug 2007 Cefixime R (disk diffusion):
24 of 146
Cefpodoxime R (disk diffusion):
31 of 146
All sensitive to ceftriaxone by disk diffusion. NGMAST ST 835 and 2180 associated with cephalosporin resistance.
Lo 200884 Hong Kong Oct 2006–Aug 2007 Ceftibuten Treatment Failure:
42 of 1228
Ceftibuten MIC90=1 (0.06–8)
Ceftriaxone MIC90=0.06 (<0.016–0.125)
Cefixime MIC90=0.125 (<0.016–0.25)
NG MAST ST 835 and 2469 associated with cephalosporin resistance.
Clendennen 1992120 Philippines September 1989 Ceftriaxone ≥0.5:
8 of 134
Cefpodoxime ≥4:
4 of 134
Clendennen 1992121 Thailand May 1990 Ceftriaxone ≥0.5:
3 of 333
Cefixime ≥4:
1 of 328
Cefpodoxime ≥4:
2 of 331
Cao 2008119 Ho Chi Minh
Ville, Vietnam
Mar 2004–Jun 2006 Ceftriaxone MIC=0.5:
1 of 121
No other cephalosporins were evaluated.
United States
Wang 2003130 Hawaii 2001 Multidrug resistance:
4 isolates
Cefixime MIC 0.25–0.5
Ceftriaxone MIC 0.125
Case report. All 3 patients with links to Asia.
Gonococcal Isolate Surveillance Project 200883 2006 1992–2006
1988–2006
Cefixime MIC 0.5–2:
48 isolates
Ceftriaxone MIC=0.5
4 isolates
Surveillance Report.

R= Resistant; LS= Less Sensitive; NG MAST= Neisseria gonorrhoeae multiple antigen sequence typing