Table 1.
| ||
---|---|---|
entry | R′ | amide (%)a |
1 | -COMe | 69 |
2 | -CO(t-Bu) | 61 |
3 | -CO(p-tolyl) | 40 |
4 | -CO(2-thienyl) | 41 |
5 | -CO(2-pyridyl) | 30 |
6 | -COC6F5 | 36 |
7 | -Me | 62 |
8 | -Ph | 60 |
Isolated yield
| ||
---|---|---|
entry | R′ | amide (%)a |
1 | -COMe | 69 |
2 | -CO(t-Bu) | 61 |
3 | -CO(p-tolyl) | 40 |
4 | -CO(2-thienyl) | 41 |
5 | -CO(2-pyridyl) | 30 |
6 | -COC6F5 | 36 |
7 | -Me | 62 |
8 | -Ph | 60 |
Isolated yield