Skip to main content
. Author manuscript; available in PMC: 2009 Apr 2.
Published in final edited form as: Org Lett. 2008 Jun 17;10(14):3005–3008. doi: 10.1021/ol8009682

Table 1.

Reaction Survey: Amidation of p-Tolylboronic Acid with O-Substituted Benzohydroxamic Acids

graphic file with name nihms98689f5.jpg
entry R′ amide (%)a
1 -COMe 69
2 -CO(t-Bu) 61
3 -CO(p-tolyl) 40
4 -CO(2-thienyl) 41
5 -CO(2-pyridyl) 30
6 -COC6F5 36
7 -Me 62
8 -Ph 60
a

Isolated yield