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. Author manuscript; available in PMC: 2010 Apr 9.
Published in final edited form as: J Med Chem. 2009 Apr 9;52(7):1943–1952. doi: 10.1021/jm801503n

Table 5.

Selectivity profile

compound p38α, IC50 (μM) Akt1, IC50 (μM) Furin, IC50 (μM) LF, IC50 (μM)
3j >100 μM 20% at 100 μM > 50 μM >100 μM
7b >100 μM 14% at 100 μM > 50 μM >100 μM
8f >100 μM 27% at 100 μM > 50 μM >100 μM
9 >100 μM 11% at 100 μM > 50 μM >100 μM