Table 3.
FEP-DW Results for Replacements of Chlorine by Hydrogen
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|---|---|---|---|---|
| Cl → H | ΔGbound (kcal/mol) | ΔΔGun (kcal/mol) | ΔΔGba (kcal/mol) | σb |
| C2 | 2.51 | 0.95 | 1.57 | 0.11 |
| C3 | 1.42 | −1.38 | 2.81 | 0.10 |
| C4 | 6.88 | 2.38 | 4.50 | 0.08 |
| C5 | 1.15 | −1.23 | 2.38 | 0.13 |
| C6 | −8.77 | −2.60 | −6.17 | 0.13 |
Computed change in free energy of binding from FEP-DW calculations.
Statistical uncertainties computed from eq 1.
