Table 6.
Summary of FEP-DW Results for Optimization of the Linker X
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|---|---|---|
| X | ΔΔGb (kcal/mol) | σ |
| CH2 | 0 | 0 |
| (R)-CHCH3 | 0.50 | 0.21 |
| (S)-CHCH3 | 2.80 | 0.18 |
| NH | 1.20 | 0.21 |
| NCH3 | −1.60 | 0.29 |
| O | 1.37 | 0.16 |
| S | −1.40 | 0.19 |
Summary of FEP-DW Results for Optimization of the Linker X
![]() | ||
|---|---|---|
| X | ΔΔGb (kcal/mol) | σ |
| CH2 | 0 | 0 |
| (R)-CHCH3 | 0.50 | 0.21 |
| (S)-CHCH3 | 2.80 | 0.18 |
| NH | 1.20 | 0.21 |
| NCH3 | −1.60 | 0.29 |
| O | 1.37 | 0.16 |
| S | −1.40 | 0.19 |