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Effect of GnRH analogues and their conjugates on cdc25 phosphatase activity
| Compound | IC50, μM
|
|
|---|---|---|
| Peptide | Conjugate | |
| MI-1544 | 1,000 | — |
| P-X-1544 | 1.33* | 0.86 |
| MI-1892 | 1,000 | — |
| P-X-1892 | 3.33* | 2.07 |
| P-X-OH | — | 37.5 |
Compounds were incubated with the enzyme as described in ref. 34.
The concentration of peptide conjugated.
