Cell penetration of MCab-Strep-Cy5 and MCab
K20A-Strep-Cy5 in wild-type and HSPG mutant CHO cells. A,
dose-dependent cell penetration of wild-type MCab-Strep-Cy5 in
wild-type and mutant CHO cells, as assessed quantitatively by FACS. Results
are from a representative experiment. The indicated concentrations are for
streptavidin-Cy5 (from 10 nm to 2.5 μm). Data were
fitted by a sigmoid equation providing the following half effective
concentrations: PC50 = 0.46 ± 0.01 μm
(wild-type CHO), 0.56 ± 0.01 μm (pgsD-677), and 0.71
± 0.01 μm (pgsB-618). a.u., absorbance units.
B, comparative cell penetration of 1 μm
MCab-Strep-Cy5 and MCab K20A-Strep-Cy5 in CHO and CHO
mutant cell lines. Results are from a representative experiment of n
= 3. Values are normalized with mean fluorescence intensity of wild-type CHO
cells.