Table I.
LmAQP1 | EC50 |
||
---|---|---|---|
[As(III)] μM | [Sb(III)] μM | [Sb(V)] μg/ml | |
vector only | 18 ± 1 | 145 ± 45 | 245 ± 40 |
wild type | 0.3 ± 0.02 | 0.4 ± 0.05 | 48 ± 4 |
E143A/E145A | 0.3 ± 0.04 | 0.4 ± 0.1 | 50 ± 5 |
E152A | 1.6 ± 0.2 | 70 ± 8 | 220 ± 50 |
E152D | 0.7 ± 0.2 | 8 ± 3 | 90 ± 6 |
E152Q | 0.3 ± 0.04 | 2.2 ± 0.7 | 65 ± 8 |
EC50 values for As(III) and Sb(III) were determined in L. donovani promastigotes transfected with wild type, E143A/E145A, E152A, E152D, E152Q LmAQP1 or vector control. Values for Sb(V) were determined for intracellular amastigotes.