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. Author manuscript; available in PMC: 2010 Apr 18.
Published in final edited form as: Tetrahedron. 2009 Apr 18;65(16):3180–3188. doi: 10.1016/j.tet.2008.11.053

Scheme 2.

Scheme 2

C- and O-arylation reactions.

(a) Aniline, pyridine, CH2Cl2; (b) Methyl iodide or ethyl iodide, K2CO3, CH3CN, 50 °C; (c) benzyl amine, Et3N, DMAP, CH2Cl2; (d) phenyl alanine methyl ester, Et3N, DMAP, CH2Cl2; (e) DIAD, PPh3, 4-buten-1-ol (f) LiAlH4, THF, 0 °C to rt.