Table 4.

Demonstration of a one-pot domino protocol.^[a]

Entry	R1	R2	R3	Product	% Yield[b]
1	H	c-C5H9	Me	7	74
2	H	c-C6H11	OH	8	86
3	4-F	Bn	OEt	9	84
4	4-F	C8H17	OH	10	90
5	H	4-ClPh	OEt	11	81
6	4-F	c-C6H11	OH	12	84
7	H	4-MeOPh	OMe	13	84

^[a]Reaction conditions: 1 (0.12 mmol), Pd₂(dba)₃·CHCl₃ (2mol-%), methyl acrylate (0.36 mmol), Bu₄NCl (0.12 mmol) in DMF at 110 °C for 14 h.

^[b]Isolated yields.