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. Author manuscript; available in PMC: 2010 Feb 17.
Published in final edited form as: Biochemistry. 2009 Feb 17;48(6):1322–1331. doi: 10.1021/bi802035f

Table 4.

Ki Values (nM) of inhibitors for CA II, CA IX mimic and CA IX

Inhibitor CA II CA IX mimic wild-type CA IX
AZM 10.1±0.7 4.9±1 3.0*
BZM 7.0±0.9 8.8±1.2 9.0±1.0
EZM < 1 < 1 -
CHL 2.0±0.4 1.1±0.2 1.0±0.3
MZM 11.8±1.8 11.4±2 9.0*
*

data from (17)