TABLE 1.
IC50 values for MLA and the AQA analogs in coapplication experiments
|
IC50
|
|||
|---|---|---|---|
| α7 | α4β2 | α3β4 | |
| μM | |||
| tPyQB | 0.13 ± 0.02 | 4.1 ± 1.0 | 1.0 ± 0.1 |
| tPy2PiB | 6.3 ± 0.6 | 86 ± 10 | 10.0 ± 1.4 |
| tkP3BzPB | 1.0 ± 0.1 | 48 ± 11 | 9.2 ± 1.2 |
| MLA | 1.2 ± 0.2 | 34 ± 5 | 2.0 ± 0.2 |
Official websites use .gov
A
.gov website belongs to an official
government organization in the United States.
Secure .gov websites use HTTPS
A lock (
) or https:// means you've safely
connected to the .gov website. Share sensitive
information only on official, secure websites.