Table 1.
Classes and specificities of HDAC inhibitors.
HDAC inhibitor | Target | |
---|---|---|
Hydroxamates | ||
TSA | Class I and II HDACs |
|
SAHA/Zolinza/vorinostat | Class I and II HDACs |
|
LAQ-824 | Class I and II HDACs |
|
LBH-589/panobinostat | Class I and II HDACs |
|
PCI 24789 | Class I and II HDACs |
|
Aliphatic acids | ||
VPA | Class I and lla HDACs |
|
Sodium Phenylbutyrate | Class I and lla HDACs |
|
Sodium Butyrate | Class I and lla HDACs |
|
Cyclic tetrapeptides | ||
Apicidin | Class I and III HDACs |
|
Trapoxin | Class I and IIa HDACs |
|
Depsipeptide/FK-228/ romidepsin |
Class IHDACs | |
Benzamides | ||
M5-275/SNDX-275 | HDAC-l, HDAC-2, HDAC-3 |
|
MGCD0103 | Class I HDACs |
SAHA: Suberoylanilide hydroxamic acid; SB: Sodium butyrate; TSA: Trichostatin A; VPA: Valproic acid.