Table 3.
Binding Constants for the Interaction of Peptides from the Long Cytoplasmic Domain of CEACAM1 with GST-β-Catenina
| Peptide | kon (M −1sec−1) | koff (sec −1) | KD (nM) |
|---|---|---|---|
| Wild type | 7.95 × 104 | 4.73 × 10−4 | 5.9 |
| K470A | 5.88 × 103 | 5.05 × 10−4 | 86 |
| H469A | 8.98 × 103 | 4.94 × 10−4 | 54 |
The GST-fusion protein (50 μg/ml) of the armadillo repeats (residues 136–671) of β-catenin was immobilized to a BIAcore CM5 chip and the binding of wild type or mutated version of the long cytoplasmic domain of CEACAM1 flowed over it vs. a CM5 chip immobilized with GST. All peptides were at 4 μM.