. Author manuscript; available in PMC: 2010 Apr 29.

Published in final edited form as: J Am Chem Soc. 2009 Apr 29;131(16):5766–5768. doi: 10.1021/ja901414u

Table 2.

Cross-coupling of primary amines and aryl iodides

ArI (1.0 equiv), amine (1.4 equiv), NaOt-Bu (1.4 equiv), 1 (0.005 – 0.2 mol%), 5 (0.005 – 0.2 mol%), toluene, 80–110 °C.

5 min reaction time.

1.0 equiv of amine was used.

Cs₂CO₃ was used as the base.