Table 4.
Percent inhibition of metabolism of a drug candidate in human liver microsomes by chemical inhibitors of CYPs
Inhibitor | Furafylline (CYP1A1/2) | Sulfaphenazole(CYP2C9) | Benzylnirvanol(CYP2C19) | Quinidine (CYP2D6) | Troleandomycin (CYP3A4) |
---|---|---|---|---|---|
Inhibition (%) | 30 | 11 | 4 | 13 | 72 |