Table 1.
Protease | Ki (nM) (Relative) inhibitor 1 | Ki (nM) (Relative) darunavir |
---|---|---|
PR | 0.27 ± 0.06 (1) | 0.34 ± 0.08 (1) |
PRD30N | 4.6 ± 0.7 (17) | 1.9 ± 0.3 (5.5) |
PRI50V | 2.1 ± 0.4 (8) | 1.3 ± 0.3 (3.9) |
PRV82A | 0.80 ± 0.06 (3) | 0.54 ± 0.04 (1.6) |
PRI84V | 0.85 ± 0.15 (3.2) | 0.56 ± 0.10 (1.7) |