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. Author manuscript; available in PMC: 2010 Sep 1.
Published in final edited form as: Bioorg Med Chem Lett. 2009 Jul 18;19(17):4967–4970. doi: 10.1016/j.bmcl.2009.07.072

Table 4.

Compound R,R′ EC50 (μM)
hmGluR44,a 		% Glu Max
2 -(CH2)4- 0.75 127
9a H,H Inactive
9b -(CH2)2- Inactive
9c -(CH2)3- Inactive
9d -(CH(CH3)2)- Inactive
9e graphic file with name nihms-140686-t0009.jpg 2.7 150
9f graphic file with name nihms-140686-t0010.jpg Inactive
9g graphic file with name nihms-140686-t0011.jpg Inactive
9h graphic file with name nihms-140686-t0012.jpg Inactive
9i graphic file with name nihms-140686-t0013.jpg inactive
9j graphic file with name nihms-140686-t0014.jpg inactive
9k graphic file with name nihms-140686-t0015.jpg 3.1 94
a

Data for inactive compounds represents the average of at least one experiment performed in triplicate; active compounds were assessed in three independent experiments in triplicate.