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. Author manuscript; available in PMC: 2010 Sep 18.
Published in final edited form as: ACS Chem Biol. 2009 Sep 18;4(9):769–781. doi: 10.1021/cb9001415

Table 1.

Peptidomimetics 4 and 1.

graphic file with name nihms144558u1.jpg
Compound 4 R1′ R2′ yield (%)a
i graphic file with name nihms144558t1.jpg graphic file with name nihms144558t2.jpg 64
j graphic file with name nihms144558t3.jpg graphic file with name nihms144558t4.jpg 74
k graphic file with name nihms144558t5.jpg graphic file with name nihms144558t6.jpg 81
l graphic file with name nihms144558t7.jpg graphic file with name nihms144558t8.jpg 98
m graphic file with name nihms144558t9.jpg graphic file with name nihms144558t10.jpg 60
n graphic file with name nihms144558t11.jpg graphic file with name nihms144558t12.jpg 68
o graphic file with name nihms144558t13.jpg graphic file with name nihms144558t14.jpg 77
p graphic file with name nihms144558t15.jpg graphic file with name nihms144558t16.jpg 78
q graphic file with name nihms144558t17.jpg graphic file with name nihms144558t18.jpg 50
r graphic file with name nihms144558t19.jpg graphic file with name nihms144558t20.jpg 40b
s graphic file with name nihms144558t21.jpg graphic file with name nihms144558t22.jpg 69b
t graphic file with name nihms144558t23.jpg graphic file with name nihms144558t24.jpg 60b
u graphic file with name nihms144558t25.jpg graphic file with name nihms144558t26.jpg 55b
v graphic file with name nihms144558t27.jpg graphic file with name nihms144558t28.jpg 84b
w graphic file with name nihms144558t29.jpg graphic file with name nihms144558t30.jpg 62b
x graphic file with name nihms144558t31.jpg graphic file with name nihms144558t32.jpg 68b
a

From intermediate 3 (see supporting) after flash chromatography.

b

After removing the side-chain benzyl protection.