TABLE 2.
Vinyl sulfone second order inhibition constants
Cruzain, ka | Rhodesain, kinact/Ki | FP-3, ka | |
---|---|---|---|
m−1 s−1 | |||
K11017 | 676,000 | 264,000 | 8,800 |
K11777 | 517,000 | 150,000 | 1,050 |
Vinyl sulfone second order inhibition constants
Cruzain, ka | Rhodesain, kinact/Ki | FP-3, ka | |
---|---|---|---|
m−1 s−1 | |||
K11017 | 676,000 | 264,000 | 8,800 |
K11777 | 517,000 | 150,000 | 1,050 |