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. Author manuscript; available in PMC: 2010 Nov 1.
Published in final edited form as: Bioorg Med Chem Lett. 2009 Sep 11;19(21):6140–6143. doi: 10.1016/j.bmcl.2009.09.015

Table 3.

Antifungal Activity of Compounds 2 and 3

IC50/MIC/MFC (µg/mL)
2 3 amphotericin B
C. neoformans 0.38/0.63/1.25 5.73/10.0/20.0 0.34/0.63/0.63
ATCC 90113
C. albicans 3.02/10.0/10.0 -a 0.26/1.25/1.25
ATCC 90028
C. krusei 1.49/2.5/2.5 -a 0.69/1.25/1.25
ATCC 6258
C. glabrata 2.67/10.0/10.0 -a 0.29/0.63/0.63
ATCC 90030
A. fumigatus 5.63/10.0/-a -a 1.02/1.25/5.0
ATCC 90906
a

not active at 20 µg/mL.